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TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018388(5,5-Bis-(3-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  2nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018350(5-(4-Methoxy-phenyl)-5-phenyl-penta-2,4-dienoic ac...)
Affinity DataIC50:  2nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018392(5-(4-Methoxy-phenyl)-5-phenyl-penta-2,4-dienoic ac...)
Affinity DataIC50:  4nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018390(5-(4-Methoxy-phenyl)-trideca-2,4-dienoic acid (1-m...)
Affinity DataIC50:  5nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018361(5-(4-Methoxy-phenyl)-undeca-2,4-dienoic acid (1-me...)
Affinity DataIC50:  9nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018349(5-(4-Methoxy-phenyl)-deca-2,4-dienoic acid (1-meth...)
Affinity DataIC50:  10nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018347(5,5-Bis-(4-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  10nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018393(5-(4-Methoxy-phenyl)-nona-2,4-dienoic acid (1-meth...)
Affinity DataIC50:  14nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018372(5-Cyclohexyl-5-(4-methoxy-phenyl)-penta-2,4-dienoi...)
Affinity DataIC50:  20nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018368(5-Cyclohexyl-5-(4-methoxy-phenyl)-penta-2,4-dienoi...)
Affinity DataIC50:  20nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018371(5,5-Bis-(3-fluoro-phenyl)-penta-2,4-dienoic acid (...)
Affinity DataIC50:  20nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018379(5-(4-Methoxy-phenyl)-hexa-2,4-dienoic acid (1-meth...)
Affinity DataIC50:  25nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018376(5,5-Bis-(3-chloro-phenyl)-penta-2,4-dienoic acid (...)
Affinity DataIC50:  25nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018356(5-(3-Fluoro-phenyl)-5-(3-methoxy-phenyl)-penta-2,4...)
Affinity DataIC50:  25nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018380(5,5-Bis-(4-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  25nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018370(5,5-Bis-(4-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  30nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018395(5-(4-Methoxy-phenyl)-penta-2,4-dienoic acid (1-met...)
Affinity DataIC50:  30nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018384(5-(4-Methoxy-phenyl)-hepta-2,4-dienoic acid (1-met...)
Affinity DataIC50:  30nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018396(5,5-Bis-(3-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  35nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018382(5,5-Bis-(4-fluoro-phenyl)-penta-2,4-dienoic acid (...)
Affinity DataIC50:  40nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018360(5-(4-Methoxy-phenyl)-6-methyl-hepta-2,4-dienoic ac...)
Affinity DataIC50:  40nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018359(5,5-Bis-(2-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  40nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018375(5-(3-Fluoro-phenyl)-5-(3-methoxy-phenyl)-penta-2,4...)
Affinity DataIC50:  40nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011671((2E,4E)-5-(4-Methoxy-phenyl)-deca-2,4-dienoic acid...)
Affinity DataIC50:  40nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018354(5-(4-Methoxy-phenyl)-octa-2,4-dienoic acid (1-meth...)
Affinity DataIC50:  50nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018394(5,5-Bis-(3,4-dimethoxy-phenyl)-penta-2,4-dienoic a...)
Affinity DataIC50:  50nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018365(6,6-Diphenyl-hexa-3,5-dienoic acid (4-pyridin-3-yl...)
Affinity DataIC50:  55nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018348(5,5-Bis-(3,4-dimethoxy-phenyl)-penta-2,4-dienoic a...)
Affinity DataIC50:  55nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018387(5,5-Bis-(4-chloro-phenyl)-penta-2,4-dienoic acid (...)
Affinity DataIC50:  60nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018386(5,5-Bis-(4-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  60nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018362(5,5-Di-p-tolyl-penta-2,4-dienoic acid (4-pyridin-3...)
Affinity DataIC50:  60nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018366(5,5-Bis-(4-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  65nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018351(5,5-Bis-(4-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  85nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018373(5,5-Diphenyl-pent-4-enoic acid (4-pyridin-3-yl-but...)
Affinity DataIC50:  100nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018389(5-Pentyl-deca-2,4-dienoic acid (1-methyl-4-pyridin...)
Affinity DataIC50:  100nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018342(5,5-Bis-(3-nitro-phenyl)-penta-2,4-dienoic acid (4...)
Affinity DataIC50:  115nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018345(5,5-Bis-(4-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  120nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018391(5,5-Bis-(3-fluoro-phenyl)-penta-2,4-dienoic acid (...)
Affinity DataIC50:  170nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)
Affinity DataIC50:  200nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018369(5,5-Bis-(4-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  200nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018352(5,5-Bis-(4-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  250nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018367(5,5-Di-p-tolyl-penta-2,4-dienoic acid (1-methyl-4-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018353(5,5-Bis-(4-fluoro-phenyl)-penta-2,4-dienoic acid (...)
Affinity DataIC50:  250nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018344(5,5-Bis-(3-fluoro-phenyl)-penta-2,4-dienoic acid (...)
Affinity DataIC50:  250nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018383(5,5-Bis-(4-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  250nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018346(5,5-Bis-(4-fluoro-phenyl)-penta-2,4-dienoic acid (...)
Affinity DataIC50:  275nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018363(5,5-Bis-(3-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  300nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018381(5,5-Bis-(4-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  300nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018358(5,5-Bis-(4-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Affinity DataIC50:  400nMAssay Description:Inhibition of [3H]-PAF binding to dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018377(5,5-Diphenyl-penta-2,4-dienoic acid (4-pyridin-3-y...)
Affinity DataIC50:  400nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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